CR4056

SKU: orb1089457

Description

CR4056 (CR 4056, CR-4056) is a novel, orally active imidazoline-2 receptor (I2R) ligand with binding IC50 of 596 nM, also selectively inhibits the enzymatic activity of MAO-A with IC50 of 202.7 nM; increases norepinephrine (NE) tissue levels both in the rat cerebral cortex and lumbar spinal cord, shows ED50 of 5.8 mg/kg in CFA rat model of inflammatory pain; shows high effectivity against bortezomib-induced painful neuropathy in rats.

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Product Categories/Products/Small Molecules,Product Categories/Products/Small Molecules/Inhibitors

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Key Properties

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CAS Number	[1004997-71-0]
MW	272.311
Formula	C₁₇H₁₂N₄
SMILES	N1=C2C(C=C(N3C=NC=C3)C=C2)=CN=C1C1=CC=CC=C1

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Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Purity:	98%
CAS Number:	1004997-71-0
MW:	272.3
Formula:	C₁₇H₁₂N₄

CR4056

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Key Properties

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CR4056 [orb1308427]

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